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2022 Update-Veterinary Drugs & Uses
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
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L1000
FAQ
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FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
procaterol 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
bronchodilators, phenethylamine derivatives
2273
72332-33-3
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
procaterol
(R,S)-Procaterol
(+/-)-Procaterol
A long-acting beta-2-adrenergic receptor agonist.
Molecular weight: 290.36
Formula: C16H22N2O3
CLOGP: 0.66
LIPINSKI: 0
HAC: 5
HDO: 4
TPSA: 81.59
ALOGS: -2.95
ROTB: 5
Drug dosage:
Dose
Unit
Route
60
mcg
Inhal.aerosol
0.10
mg
O
ADMET properties:
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Property
Value
Reference
BA (Bioavailability)
40 %
Kim MT, Sedykh A, Chakravarti SK, Saiakhov RD, Zhu H
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Approvals:
None
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
R03AC16
RESPIRATORY SYSTEM
DRUGS FOR OBSTRUCTIVE AIRWAY DISEASES
ADRENERGICS, INHALANTS
Selective beta-2-adrenoreceptor agonists
ATC
R03CC08
RESPIRATORY SYSTEM
DRUGS FOR OBSTRUCTIVE AIRWAY DISEASES
ADRENERGICS FOR SYSTEMIC USE
Selective beta-2-adrenoreceptor agonists
MeSH PA
D018663
Adrenergic Agents
MeSH PA
D000322
Adrenergic Agonists
MeSH PA
D058666
Adrenergic beta-2 Receptor Agonists
MeSH PA
D000318
Adrenergic beta-Agonists
MeSH PA
D018927
Anti-Asthmatic Agents
MeSH PA
D001993
Bronchodilator Agents
MeSH PA
D018377
Neurotransmitter Agents
MeSH PA
D018373
Peripheral Nervous System Agents
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
None
🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
10.58
acidic
pKa2
11.26
acidic
pKa3
9.7
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Beta-2 adrenergic receptor
GPCR
P07550
ADRB2_HUMAN
AGONIST
EC50
8.43
IUPHAR
IUPHAR
D(2) dopamine receptor
GPCR
P14416
DRD2_HUMAN
Ki
4.07
CHEMBL
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External reference:
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ID
Source
003878
NDDF
34530
RXNORM
3464
IUPHAR_LIGAND_ID
4259
INN_ID
4916
PUBCHEM_CID
703566006
SNOMEDCT_US
C0072032
UMLSCUI
CHEBI:135209
CHEBI
CHEMBL160519
ChEMBL_ID
D017265
MESH_DESCRIPTOR_UI
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Pharmaceutical products:
None
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procaterol