DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
Scroll
All
FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
carmofur 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
uridine derivatives used as antiviral agents and as antineoplastics
511
61422-45-5
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
1-hexylcarbamoyl-5-fluorouracil
carmofur
mifurol
yamaful
Molecular weight: 257.27
Formula: C11H16FN3O3
CLOGP: 2.55
LIPINSKI: 0
HAC: 6
HDO: 2
TPSA: 78.51
ALOGS: -3.72
ROTB: 5
Drug dosage:
None
ADMET properties:
None
Approvals:
None
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
Show
10
25
50
100
entries
Search:
Source
Code
Description
ATC
L01BC04
ANTINEOPLASTIC AND IMMUNOMODULATING AGENTS
ANTINEOPLASTIC AGENTS
ANTIMETABOLITES
Pyrimidine analogues
MeSH PA
D000970
Antineoplastic Agents
Showing 1 to 2 of 2 entries
Previous
1
Next
Drug Use
| Suggest Off label Use Form|
|View source of the data|
Show
10
25
50
100
entries
Search:
Disease
Relation
SNOMED_ID
DOID
Malignant tumor of colon
indication
363406005
DOID:219
Showing 1 to 1 of 1 entries
Previous
1
Next
🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
Show
10
25
50
100
entries
Search:
Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
6.55
acidic
pKa2
13.95
acidic
Showing 1 to 2 of 2 entries
Previous
1
Next
Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
Show
10
25
50
100
entries
Search:
Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Cytochrome P450 2D6
Enzyme
P10635
CP2D6_HUMAN
IC50
5.30
DRUG MATRIX
Mitogen-activated protein kinase 3
Kinase
P27361
MK03_HUMAN
IC50
5.21
DRUG MATRIX
Acid ceramidase
Enzyme
Q13510
ASAH1_HUMAN
IC50
7.68
CHEMBL
Sulfide:quinone oxidoreductase, mitochondrial
Unclassified
Q9Y6N5
SQRD_HUMAN
IC50
4.70
CHEMBL
Fatty-acid amide hydrolase 1
Enzyme
FAAH1_RAT
IC50
7.60
CHEMBL
Acid ceramidase
Enzyme
ASAH1_RAT
IC50
7.54
CHEMBL
Replicase polyprotein 1ab
Enzyme
R1AB_SARS2
IC50
5.74
CHEMBL
Showing 1 to 7 of 7 entries
Previous
1
Next
External reference:
Show
10
25
50
100
entries
Search:
ID
Source
010893
NDDF
2577
PUBCHEM_CID
5042
INN_ID
C0044401
UMLSCUI
C017367
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:31360
CHEBI
CHEMBL460499
ChEMBL_ID
D01784
KEGG_DRUG
DB09010
DRUGBANK_ID
HA82M3RAB2
UNII
Showing 1 to 10 of 10 entries
Previous
1
Next
Pharmaceutical products:
None
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
carmofur