bazedoxifene 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
antiestrogens or estrogen receptor modulators, clomifene and tamoxifen derivatives 4334 198481-32-2

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • TSE424
  • TSE-424
  • bazedoxifene acetate
  • bazedoxifene
  • conbriza
an estrogen agonist/antagonist that acts as an agonist in some estrogen-sensitive tissues and an antagonist in others
  • Molecular weight: 470.61
  • Formula: C30H34N2O3
  • CLOGP: 7.15
  • LIPINSKI: 1
  • HAC: 5
  • HDO: 2
  • TPSA: 57.86
  • ALOGS: -5.92
  • ROTB: 7
  • Status: OFP
    • Legend:
    OFP - off patent
    OFM - off market
    ONP - on patent

Drug dosage:

DoseUnitRoute
20 mg O

ADMET properties:

Approvals:

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

Drug Use | Suggest Off label Use Form| |View source of the data|




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Orange Book patent data (new drug applications)

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

External reference:

Pharmaceutical products:

bazedoxifene