ormeloxifene 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
antiestrogens or estrogen receptor modulators, clomifene and tamoxifen derivatives 570 31477-60-8

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • centchroman
  • ormeloxifene
  • ormeloxifen
  • centron
A non-steroidal anti-fertility agent with anti-hormonal properties.
  • Molecular weight: 457.61
  • Formula: C30H35NO3
  • CLOGP: 7.54
  • LIPINSKI: 1
  • HAC: 4
  • HDO: 0
  • TPSA: 30.93
  • ALOGS: -6.65
  • ROTB: 7

Drug dosage:

None

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

SourceCodeDescription
ATC G03XC04 GENITO URINARY SYSTEM AND SEX HORMONES
SEX HORMONES AND MODULATORS OF THE GENITAL SYSTEM
OTHER SEX HORMONES AND MODULATORS OF THE GENITAL SYSTEM
Selective estrogen receptor modulators
MeSH PA D003270 Contraceptive Agents
MeSH PA D003271 Contraceptive Agents, Female
MeSH PA D003283 Contraceptives, Postcoital, Synthetic
MeSH PA D004965 Estrogen Antagonists
MeSH PA D006727 Hormone Antagonists
MeSH PA D012102 Reproductive Control Agents

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 8.9 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

IDSource
D08301 KEGG_DRUG
C0007665 UMLSCUI
CHEBI:135742 CHEBI
CHEMBL154126 ChEMBL_ID
DB13310 DRUGBANK_ID
C508548 MESH_SUPPLEMENTAL_RECORD_UI
7100 INN_ID
44AXY5VE90 UNII
35805 PUBCHEM_CID
1187476007 SNOMEDCT_US
1187495000 SNOMEDCT_US
D002486 MESH_DESCRIPTOR_UI

Pharmaceutical products:

None