bezitramide 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
363 15301-48-1

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • R-4845
  • bezitramide monohydrochloride
  • bezitramide hydrochloride
  • bezitramide HCl
  • bezitramide
  • benzitramide
  • burgodin
  • Molecular weight: 492.62
  • Formula: C31H32N4O2
  • CLOGP: 5.28
  • LIPINSKI: 1
  • HAC: 6
  • HDO: 0
  • TPSA: 67.65
  • ALOGS: -4.87
  • ROTB: 7

Drug dosage:

DoseUnitRoute
15 mg O

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

SourceCodeDescription
ATC N02AC05 NERVOUS SYSTEM
ANALGESICS
OPIOIDS
Diphenylpropylamine derivatives
MeSH PA D000700 Analgesics
MeSH PA D002491 Central Nervous System Agents
MeSH PA D018373 Peripheral Nervous System Agents
MeSH PA D018689 Sensory System Agents

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 6.65 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

IDSource
D07289 KEGG_DRUG
59708-44-0 SECONDARY_CAS_RN
C0053535 UMLSCUI
CHEBI:135794 CHEBI
CHEMBL2104149 ChEMBL_ID
DB01459 DRUGBANK_ID
C004461 MESH_SUPPLEMENTAL_RECORD_UI
1942 INN_ID
3KXW0Y310I UNII
61791 PUBCHEM_CID

Pharmaceutical products:

None