DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
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L1000
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FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
imidafenacin 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
muscarinic receptors antagonists
4902
170105-16-5
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
imidafenacin
uritos
KRP-197
KRP 197
Molecular weight: 319.41
Formula: C20H21N3O
CLOGP: 2.23
LIPINSKI: 0
HAC: 4
HDO: 1
TPSA: 60.91
ALOGS: -4.53
ROTB: 6
Drug dosage:
None
ADMET properties:
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Property
Value
Reference
CL (Clearance)
6.10 mL/min/kg
Lombardo F, Berellini G, Obach RS
t_half (Half-life)
3.20 hours
Lombardo F, Berellini G, Obach RS
Vd (Volume of distribution)
1.51 L/kg
Lombardo F, Berellini G, Obach RS
BA (Bioavailability)
0.58 %
Kawashima H, Watanabe R, Esaki T, Kuroda M, Nagao C, Natsume-Kitatani Y, Ohashi R, Komura H, Mizuguchi K
fu (Fraction unbound in plasma)
0.12 %
Lombardo F, Berellini G, Obach RS
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Approvals:
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Date
Agency
Company
Orphan
April 18, 2007
PMDA
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
G04BD14
GENITO URINARY SYSTEM AND SEX HORMONES
UROLOGICALS
UROLOGICALS
Drugs for urinary frequency and incontinence
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Bladder muscle dysfunction - overactive
indication
236633002
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
13.68
acidic
pKa2
6.35
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Muscarinic acetylcholine receptor M3
GPCR
P20309
ACM3_HUMAN
ANTAGONIST
Kb
9.50
SCIENTIFIC LITERATURE
SCIENTIFIC LITERATURE
Muscarinic acetylcholine receptor M1
GPCR
P11229
ACM1_HUMAN
Kb
8.38
SCIENTIFIC LITERATURE
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External reference:
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ID
Source
6433090
PUBCHEM_CID
8402
INN_ID
C120953
MESH_SUPPLEMENTAL_RECORD_UI
C1876226
UMLSCUI
CHEBI:134720
CHEBI
CHEMBL53366
ChEMBL_ID
D06273
KEGG_DRUG
DB09262
DRUGBANK_ID
XJR8Y07LJO
UNII
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Pharmaceutical products:
None
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imidafenacin