azidocillin 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
antibiotics, 6-aminopenicillanic acid derivatives 273 17243-38-8

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • azidocillin potasium
  • azidocillin sodium
  • azidocillin
  • azidobenzylpenicillin
antibiotic similir to ampicillin; minor descriptor (75-86); on line & INDEX MEDICUS search PENICILLIN G/AA (75-86); RN given refers to (2S-(2alpha,5alpha,6beta(S*))-isomer)
  • Molecular weight: 375.40
  • Formula: C16H17N5O4S
  • CLOGP: 2.60
  • LIPINSKI: 0
  • HAC: 9
  • HDO: 2
  • TPSA: 116.14
  • ALOGS: -2.79
  • ROTB: 5

Drug dosage:

DoseUnitRoute
1.50 g O

ADMET properties:

PropertyValueReference
BA (Bioavailability) 60 % Kim MT, Sedykh A, Chakravarti SK, Saiakhov RD, Zhu H

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

SourceCodeDescription
ATC J01CE04 ANTIINFECTIVES FOR SYSTEMIC USE
ANTIBACTERIALS FOR SYSTEMIC USE
BETA-LACTAM ANTIBACTERIALS, PENICILLINS
Beta-lactamase sensitive penicillins

Drug Use | Suggest Off label Use Form| |View source of the data|

DiseaseRelationSNOMED_IDDOID
Respiratory tract infection indication 275498002




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 2.79 acidic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

IDSource
D07235 KEGG_DRUG
35334-12-4 SECONDARY_CAS_RN
18609 RXNORM
C0052772 UMLSCUI
CHEBI:51758 CHEBI
CHEMBL2105907 ChEMBL_ID
DB08795 DRUGBANK_ID
C100243 MESH_SUPPLEMENTAL_RECORD_UI
15574941 PUBCHEM_CID
12291 IUPHAR_LIGAND_ID
2458 INN_ID
R8XDP7L3SL UNII
006819 NDDF
006820 NDDF

Pharmaceutical products:

None