sulfisomidine 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definition	Drug id	CAS RN
anti-infectives, sulfonamides	2526	515-64-0

Description:

Molecule

Description

Molfile Inchi Smiles

Synonyms:

sulfasomidine
sulfadimetine
sulfaisodimerazine
sulfamethine
sulfasomidin
sulfisomidin
sulfisomidine
sulphasomidine
sulphisomidine
sulfaisodimidine

A sulfanilamide antibacterial agent.

Molecular weight: 278.33
Formula: C12H14N4O2S
CLOGP: 1.10
LIPINSKI: 0
HAC: 6
HDO: 2
TPSA: 97.97
ALOGS: -3.09
ROTB: 2

Drug dosage:

Dose	Unit	Route
4	g	O
4	g	P

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

Source	Code	Description
ATC	J01EB01	ANTIINFECTIVES FOR SYSTEMIC USE ANTIBACTERIALS FOR SYSTEMIC USE SULFONAMIDES AND TRIMETHOPRIM Short-acting sulfonamides
MeSH PA	D000890	Anti-Infective Agents
CHEBI has role	CHEBI:35441	antiinfective agents

Drug Use | Suggest Off label Use Form| |View source of the data|

None

🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation level	Dissociation constant	Type (acidic/basic)
pKa1	7.21	acidic
pKa2	4.49	Basic
pKa3	2.24	Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

Target	Class	Pharos	UniProt	Action	Type	Activity value (-log[M])	Mechanism action	Bioact source	MoA source
Protein argonaute-2	Unclassified	Q9UKV8	AGO2_HUMAN		Kd	5.37		CHEMBL

External reference:

ID	Source
N0000166865	NUI
D01526	KEGG_DRUG
CHEBI:32166	CHEBI
CHEMBL485696	ChEMBL_ID
99	INN_ID
DB13283	DRUGBANK_ID
W03L3ODK6E	UNII
10206	RXNORM
002823	NDDF
4014000	SNOMEDCT_US
C0038744	UMLSCUI
D013443	MESH_DESCRIPTOR_UI
5343	PUBCHEM_CID

Pharmaceutical products:

None