DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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Structure 🔎
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
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All
FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
anecortave 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
corticosteroids, except prednisolone derivatives
217
7753-60-8
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
anecortave acetate
anecortave
retaane
Molecular weight: 386.49
Formula: C23H30O5
CLOGP: 2.87
LIPINSKI: 0
HAC: 5
HDO: 1
TPSA: 80.67
ALOGS: -4.53
ROTB: 4
Drug dosage:
None
ADMET properties:
None
Approvals:
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Date
Agency
Company
Orphan
Jan. 1, 2006
YEAR INTRODUCED
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
S01LA02
SENSORY ORGANS
OPHTHALMOLOGICALS
OCULAR VASCULAR DISORDER AGENTS
Antineovascularisation agents
MeSH PA
D020533
Angiogenesis Inhibitors
MeSH PA
D000970
Antineoplastic Agents
MeSH PA
D006131
Growth Inhibitors
MeSH PA
D006133
Growth Substances
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Exudative age-related macular degeneration
indication
414173003
DOID:10873
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
12.5
acidic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Plasminogen activator inhibitor 1
Secreted
P05121
PAI1_HUMAN
WOMBAT-PK
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External reference:
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entries
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ID
Source
011285
NDDF
011286
NDDF
10184-70-0
SECONDARY_CAS_RN
7074810
PUBCHEM_CID
7747
INN_ID
C108424
MESH_SUPPLEMENTAL_RECORD_UI
C1693912
UMLSCUI
C418047
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:31215
CHEBI
CHEMBL2106613
ChEMBL_ID
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Pharmaceutical products:
None
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anecortave