DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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Structure 🔎
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
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FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
nadifloxacin 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
antibacterials, nalidixic acid derivatives
1864
124858-35-1
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
OPC 7251
OPC-7251
nadixa
jinofloxacin
nadifloxacin
(R)-isomer does not induce chromosomal aberrations, unlike (S)-isomer; structure given in first source
Molecular weight: 360.39
Formula: C19H21FN2O4
CLOGP: 1.66
LIPINSKI: 0
HAC: 6
HDO: 2
TPSA: 81.08
ALOGS: -2.76
ROTB: 2
Drug dosage:
None
ADMET properties:
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Property
Value
Reference
t_half (Half-life)
6.04 hours
Lombardo F, Berellini G, Obach RS
CL (Clearance)
0.54 mL/min/kg
Lombardo F, Berellini G, Obach RS
Vd (Volume of distribution)
0.25 L/kg
Lombardo F, Berellini G, Obach RS
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Approvals:
None
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
D10AF05
DERMATOLOGICALS
ANTI-ACNE PREPARATIONS
ANTI-ACNE PREPARATIONS FOR TOPICAL USE
Antiinfectives for treatment of acne
CHEBI has role
CHEBI:36047
antibacterial drugs
MeSH PA
D000900
Anti-Bacterial Agents
MeSH PA
D000890
Anti-Infective Agents
MeSH PA
D000970
Antineoplastic Agents
MeSH PA
D004791
Enzyme Inhibitors
MeSH PA
D059005
Topoisomerase II Inhibitors
MeSH PA
D059003
Topoisomerase Inhibitors
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Acne vulgaris
indication
88616000
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
6.03
acidic
pKa2
3.1
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
None
External reference:
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ID
Source
007854
NDDF
4410
PUBCHEM_CID
6702
INN_ID
698260001
SNOMEDCT_US
6CL9Y5YZEQ
UNII
C0286402
UMLSCUI
C062127
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:31889
CHEBI
CHEMBL363449
ChEMBL_ID
D01147
KEGG_DRUG
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Pharmaceutical products:
None
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nadifloxacin