phenazone 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
anti-inflammatory analgesics, phenylbutazone derivatives 861 60-80-0

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • phenazone
  • analgesin
  • analgesine
  • anodynine
  • antipyrin
  • azophen
  • azophene
  • dimethyloxychinizin
  • dimethyloxyquinazine
  • fenazone
  • methozin
  • oxydimethylquinazine
  • phenazon
  • pyrazophyl
  • phenylone
  • antipyrine
An analgesic and antipyretic that has been given by mouth and as ear drops. Antipyrine is often used in testing the effects of other drugs or diseases on drug-metabolizing enzymes in the liver. (From Martindale, The Extra Pharmacopoeia, 30th ed, p29)
  • Molecular weight: 188.23
  • Formula: C11H12N2O
  • CLOGP: 0.19
  • LIPINSKI: 0
  • HAC: 3
  • HDO: 0
  • TPSA: 23.55
  • ALOGS: -0.60
  • ROTB: 1

Drug dosage:

DoseUnitRoute
3 g O
3 g O

ADMET properties:

Approvals:

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

Drug Use | Suggest Off label Use Form| |View source of the data|




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

None

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

External reference:

Pharmaceutical products:

phenazone