DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
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L1000
FAQ
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FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
beclabuvir 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
antivirals RNA polymerase (NS5B) inhibitors
5215
958002-33-0
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
beclabuvir
beclabuvir hydrochloride
beclabuvir HCl
BMS-791325
BMS 791325
an NS5B inhibitor and antiviral agent
Molecular weight: 659.85
Formula: C36H45N5O5S
CLOGP: 6.20
LIPINSKI: 2
HAC: 10
HDO: 1
TPSA: 104.19
ALOGS: -5.19
ROTB: 4
Drug dosage:
None
ADMET properties:
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Property
Value
Reference
t_half (Half-life)
5.38 hours
Lombardo F, Berellini G, Obach RS
CL (Clearance)
1.33 mL/min/kg
Lombardo F, Berellini G, Obach RS
Vd (Volume of distribution)
0.50 L/kg
Lombardo F, Berellini G, Obach RS
fu (Fraction unbound in plasma)
0.01 %
Lombardo F, Berellini G, Obach RS
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Approvals:
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Date
Agency
Company
Orphan
Dec. 19, 2016
PMDA
Bristol-Myers Squibb
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
J05AP58
ANTIINFECTIVES FOR SYSTEMIC USE
ANTIVIRALS FOR SYSTEMIC USE
DIRECT ACTING ANTIVIRALS
Antivirals for treatment of HCV infections
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Chronic hepatitis C
indication
128302006
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
3.9
acidic
pKa2
8.35
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Potassium voltage-gated channel subfamily H member 2
Ion channel
Q12809
KCNH2_HUMAN
IC50
4.61
CHEMBL
NS5B protein
Enzyme
Q8JXU8_9HEPC
IC50
6.72
CHEMBL
RNA-directed RNA polymerase
Unclassified
O39930_9HEPC
IC50
6.72
CHEMBL
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External reference:
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ID
Source
56934415
PUBCHEM_CID
958002-36-3
SECONDARY_CAS_RN
9899
INN_ID
C4045497
UMLSCUI
C587012
MESH_SUPPLEMENTAL_RECORD_UI
CHEMBL3126842
ChEMBL_ID
CHEMBL3137325
ChEMBL_ID
D10611
KEGG_DRUG
DB12225
DRUGBANK_ID
MYW1X5CO9S
UNII
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Pharmaceutical products:
None
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beclabuvir