buserelin ๐Ÿถ Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
pituitary hormone-release stimulating peptides 436 57982-77-1

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • buserelin
  • etilamide
  • receptal
  • buserelin acetate
  • suprecur
A potent synthetic analog of GONADOTROPIN-RELEASING HORMONE with D-serine substitution at residue 6, glycine10 deletion, and other modifications.
  • Molecular weight: 1239.45
  • Formula: C60H86N16O13
  • CLOGP: -3.63
  • LIPINSKI: 3
  • HAC: 29
  • HDO: 16
  • TPSA: 438.27
  • ALOGS: -4.51
  • ROTB: 33

Drug dosage:

DoseUnitRoute
0.11 mg implant
1.20 mg N
1.50 mg P

ADMET properties:

Approvals:

FDA Adverse Event Reporting System (Female)

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

Drug Use | Suggest Off label Use Form| |View source of the data|




๐Ÿถ Veterinary Drug Use

None

๐Ÿถ Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

External reference:

Pharmaceutical products:

None

buserelin