chlorthenoxazine 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
3707 132-89-8

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • chlorthenoxazine
  • apirazin
  • chlorethylbenzmethoxazone
  • ossapirina
  • ossazone
  • piroxina
  • reumagrip
  • valmorin
  • Molecular weight: 211.65
  • Formula: C10H10ClNO2
  • CLOGP: 1.55
  • LIPINSKI: 0
  • HAC: 3
  • HDO: 1
  • TPSA: 38.33
  • ALOGS: -2.16
  • ROTB: 2

Drug dosage:

None

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

None

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 12.97 acidic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

TargetClassPharosUniProtActionTypeActivity value
(-log[M])		Mechanism
action		Bioact sourceMoA source
Poly [ADP-ribose] polymerase 1 Enzyme IC50 5.07 CHEMBL

External reference:

IDSource
KA0B657LV3 UNII
C0055478 UMLSCUI
CHEBI:134882 CHEBI
CHEMBL124815 ChEMBL_ID
8602 PUBCHEM_CID
962 INN_ID
20891 RXNORM
004336 NDDF

Pharmaceutical products:

None