tocainide 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
Class I antiarrhythmics, procainamide and lidocaine derivatives 2686 41708-72-9

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • tocainide hydrochloride
  • tocainide
  • (RS)-Tocainide
  • (+/-)-Tocainide
  • DL-Tocainide
  • tocainide HCl
An antiarrhythmic agent which exerts a potential- and frequency-dependent block of SODIUM CHANNELS.
  • Molecular weight: 192.26
  • Formula: C11H16N2O
  • CLOGP: 0.26
  • LIPINSKI: 0
  • HAC: 3
  • HDO: 2
  • TPSA: 55.12
  • ALOGS: -2.08
  • ROTB: 2

  • Status: OFM

  • Legend:
    OFP - off patent
    OFM - off market
    ONP - on patent

Drug dosage:

DoseUnitRoute
1.20 g O
1.20 g P

ADMET properties:

Approvals:

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

Drug Use | Suggest Off label Use Form| |View source of the data|




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

External reference:

Pharmaceutical products:

None

tocainide