tilbroquinol 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
quinoline derivatives 2662 7175-09-9

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • tilbroquinol
  • 5-Methyl-7-bromo-8-hydroxyquinoline
  • Molecular weight: 238.08
  • Formula: C10H8BrNO
  • CLOGP: 3.28
  • LIPINSKI: 0
  • HAC: 2
  • HDO: 1
  • TPSA: 33.12
  • ALOGS: -2.90
  • ROTB: 0

Drug dosage:

None

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

SourceCodeDescription
ATC P01AA05 ANTIPARASITIC PRODUCTS, INSECTICIDES AND REPELLENTS
ANTIPROTOZOALS
AGENTS AGAINST AMOEBIASIS AND OTHER PROTOZOAL DISEASES
Hydroxyquinoline derivatives
ATC P01AA30 ANTIPARASITIC PRODUCTS, INSECTICIDES AND REPELLENTS
ANTIPROTOZOALS
AGENTS AGAINST AMOEBIASIS AND OTHER PROTOZOAL DISEASES
Hydroxyquinoline derivatives

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 8.74 acidic
pKa2 3.6 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

IDSource
D07351 KEGG_DRUG
C0618388 UMLSCUI
CHEBI:134965 CHEBI
CHEMBL1788385 ChEMBL_ID
DB13222 DRUGBANK_ID
65592 PUBCHEM_CID
C037665 MESH_SUPPLEMENTAL_RECORD_UI
5008 INN_ID
P6SB125NHA UNII
166718 RXNORM
005354 NDDF
735058009 SNOMEDCT_US

Pharmaceutical products:

None