astemizole 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
antihistaminics 249 68844-77-9

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • R 43 512
  • astemizole
  • astemisan
  • hismanal
  • histazol
Antihistamine drug now withdrawn from the market in many countries because of rare but potentially fatal side effects.
  • Molecular weight: 458.58
  • Formula: C28H31FN4O
  • CLOGP: 5.84
  • LIPINSKI: 1
  • HAC: 5
  • HDO: 1
  • TPSA: 42.32
  • ALOGS: -5.58
  • ROTB: 8

Drug dosage:

DoseUnitRoute
10 mg O

ADMET properties:

Approvals:

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

Drug Use | Suggest Off label Use Form| |View source of the data|




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

External reference:

Pharmaceutical products:

None

astemizole