DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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Structure 🔎
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L1000
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FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
quinupramine 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
substances of the imipramine group
2348
31721-17-2
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
quinupramine monohydrochloride
quinupramine hydrochloride
quinupramine HCl
quinupramine tartrate
quinupramine
kevopril
kinupril
Molecular weight: 304.44
Formula: C21H24N2
CLOGP: 4.78
LIPINSKI: 0
HAC: 2
HDO: 0
TPSA: 6.48
ALOGS: -4.24
ROTB: 1
Drug dosage:
None
ADMET properties:
None
Approvals:
None
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
N06AA23
NERVOUS SYSTEM
PSYCHOANALEPTICS
ANTIDEPRESSANTS
Non-selective monoamine reuptake inhibitors
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
None
🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
8.15
Basic
pKa2
5.01
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
None
External reference:
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ID
Source
005341
NDDF
29O61HFF4L
UNII
35242
RXNORM
3697
INN_ID
93154
PUBCHEM_CID
C0072896
UMLSCUI
C028338
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:135292
CHEBI
CHEMBL107360
ChEMBL_ID
D07336
KEGG_DRUG
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Pharmaceutical products:
None
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quinupramine