DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
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L1000
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FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
quinagolide 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
dopamine receptor agonists, ergoline derivatives
2339
87056-78-8
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
quinagolide
norprolac
Molecular weight: 395.56
Formula: C20H33N3O3S
CLOGP: 3.73
LIPINSKI: 0
HAC: 6
HDO: 2
TPSA: 72.88
ALOGS: -3.41
ROTB: 5
Drug dosage:
Dose
Unit
Route
75
mcg
O
ADMET properties:
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Property
Value
Reference
BA (Bioavailability)
99 %
Kim MT, Sedykh A, Chakravarti SK, Saiakhov RD, Zhu H
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Approvals:
None
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
G02CB04
GENITO URINARY SYSTEM AND SEX HORMONES
OTHER GYNECOLOGICALS
OTHER GYNECOLOGICALS
Prolactine inhibitors
MeSH PA
D015259
Dopamine Agents
MeSH PA
D018491
Dopamine Agonists
MeSH PA
D018377
Neurotransmitter Agents
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
None
🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
10.45
acidic
pKa2
11.15
acidic
pKa3
8.35
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Serotonin (5-HT) receptor
GPCR
5HT2C_RAT
5HT2A_RAT
5HT1A_RAT
5HT1B_RAT
5HT1D_RAT
5HT1F_RAT
5HT2B_RAT
5HT6R_RAT
5HT7R_RAT
5HT5A_RAT
5HT5B_RAT
5HT3A_RAT
5HT4R_RAT
5HT3B_RAT
IC50
5.64
CHEMBL
Adrenergic receptor alpha-2
GPCR
ADA2B_RAT
ADA2C_RAT
ADA2A_RAT
IC50
5.25
CHEMBL
Dopamine receptor
GPCR
DRD2_BOVIN
DRD1_BOVIN
IC50
7.72
CHEMBL
Adrenergic receptor alpha-1
GPCR
ADA1B_RAT
ADA1D_RAT
ADA1A_RAT
IC50
5.22
CHEMBL
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External reference:
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ID
Source
005470
NDDF
152131
RXNORM
3086400
PUBCHEM_CID
326066005
SNOMEDCT_US
395850005
SNOMEDCT_US
6545
INN_ID
80Q9QWN15M
UNII
C0256089
UMLSCUI
C046650
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:135627
CHEBI
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Pharmaceutical products:
None
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quinagolide