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2022 Update-Veterinary Drugs & Uses
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
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L1000
FAQ
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All
FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
lornoxicam 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
anti-inflammatory, isoxicam derivatives
1609
70374-39-9
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
lornoxicam
chlortenoxicam
lorcam
xefocam
Molecular weight: 371.81
Formula: C13H10ClN3O4S2
CLOGP: 2.34
LIPINSKI: 0
HAC: 7
HDO: 2
TPSA: 99.60
ALOGS: -3.93
ROTB: 2
Drug dosage:
Dose
Unit
Route
12
mg
O
12
mg
P
12
mg
R
ADMET properties:
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Property
Value
Reference
BA (Bioavailability)
1 %
Kawashima H, Watanabe R, Esaki T, Kuroda M, Nagao C, Natsume-Kitatani Y, Ohashi R, Komura H, Mizuguchi K
Vd (Volume of distribution)
0.14 L/kg
Kawashima H, Watanabe R, Esaki T, Kuroda M, Nagao C, Natsume-Kitatani Y, Ohashi R, Komura H, Mizuguchi K
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Approvals:
None
FDA Adverse Event Reporting System (Female)
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MedDRA adverse event term
Likelihood ratio
Likelihood ratio threshold
Patients taking drug having adverse event
Patients taking drug not having adverse event
Patients not taking drug having adverse event
Patients not taking drug not having adverse event
Angioedema
56.68
52.86
18
373
47947
63440684
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FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
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MedDRA adverse event term
Likelihood ratio
Likelihood ratio threshold
Patients taking drug having adverse event
Patients taking drug not having adverse event
Patients not taking drug having adverse event
Patients not taking drug not having adverse event
Drug interaction
46.11
38.17
34
669
415149
79328536
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FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
M01AC05
MUSCULO-SKELETAL SYSTEM
ANTIINFLAMMATORY AND ANTIRHEUMATIC PRODUCTS
ANTIINFLAMMATORY AND ANTIRHEUMATIC PRODUCTS, NON-STEROIDS
Oxicams
CHEBI has role
CHEBI:35475
non-steroidal anti-inflammatory agent
CHEBI has role
CHEBI:35493
anti-pyretic
MeSH PA
D000700
Analgesics
MeSH PA
D018712
Analgesics, Non-Narcotic
MeSH PA
D000893
Anti-Inflammatory Agents
MeSH PA
D000894
Anti-Inflammatory Agents, Non-Steroidal
MeSH PA
D018501
Antirheumatic Agents
MeSH PA
D018373
Peripheral Nervous System Agents
MeSH PA
D018689
Sensory System Agents
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Pain
indication
22253000
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
0.98
acidic
pKa2
8.43
acidic
pKa3
5.18
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
None
External reference:
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ID
Source
007785
NDDF
20890
RXNORM
391655005
SNOMEDCT_US
412013008
SNOMEDCT_US
54690031
PUBCHEM_CID
6233
INN_ID
C0055477
UMLSCUI
C059451
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:31783
CHEBI
CHEMBL1569487
ChEMBL_ID
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Pharmaceutical products:
None
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lornoxicam