DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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Structure 🔎
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
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All
FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
gliquidone 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
antihyperglycaemics
1302
33342-05-1
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
gliquidone
glurenorm
beglynor
gliquidone calcium
gliquidone monosodium
gliquidone sodium
Molecular weight: 527.64
Formula: C27H33N3O6S
CLOGP: 5.06
LIPINSKI: 2
HAC: 9
HDO: 2
TPSA: 121.88
ALOGS: -5.38
ROTB: 6
Drug dosage:
Dose
Unit
Route
60
mg
O
ADMET properties:
None
Approvals:
None
FDA Adverse Event Reporting System (Female)
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MedDRA adverse event term
Likelihood ratio
Likelihood ratio threshold
Patients taking drug having adverse event
Patients taking drug not having adverse event
Patients not taking drug having adverse event
Patients not taking drug not having adverse event
Stevens-Johnson syndrome
77.34
74.77
19
296
24931
63463776
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FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
A10BB08
ALIMENTARY TRACT AND METABOLISM
DRUGS USED IN DIABETES
BLOOD GLUCOSE LOWERING DRUGS, EXCL. INSULINS
Sulfonylureas
MeSH PA
D007004
Hypoglycemic Agents
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Diabetes mellitus type 2
indication
44054006
DOID:9352
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
5.31
acidic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Sulfonylurea receptor 1, Kir6.2
Ion channel
Q09428
Q14654
ABCC8_HUMAN
KCJ11_HUMAN
BLOCKER
Kd
9
SCIENTIFIC LITERATURE
SCIENTIFIC LITERATURE
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External reference:
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ID
Source
003974
NDDF
25793
RXNORM
325249006
SNOMEDCT_US
3308
INN_ID
395732008
SNOMEDCT_US
91610
PUBCHEM_CID
C0061328
UMLSCUI
C010969
MESH_SUPPLEMENTAL_RECORD_UI
C7C2QDD75P
UNII
CHEBI:93416
CHEBI
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Pharmaceutical products:
None
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gliquidone