zolazepam 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
diazepam derivatives 5647 31352-82-6

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • zolazepam
  • zolazepam hydrochloride
A pyrazolodiazepinone with pharmacological actions similar to ANTI-ANXIETY AGENTS. It is commonly used in combination with TILETAMINE to obtain immobilization and anesthesia in animals
  • Molecular weight: 286.31
  • Formula: C15H15FN4O
  • CLOGP: 0.63
  • LIPINSKI: 0
  • HAC: 5
  • HDO: 0
  • TPSA: 50.49
  • ALOGS: -3.03
  • ROTB: 1

Drug dosage:

None

ADMET properties:

None

Approvals:

DateAgencyCompanyOrphan
None FDA

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

SourceCodeDescription
MeSH PA D014151 Anti-Anxiety Agents
MeSH PA D002491 Central Nervous System Agents
MeSH PA D002492 Central Nervous System Depressants
MeSH PA D018682 GABA Agents
MeSH PA D018757 GABA Modulators
MeSH PA D018377 Neurotransmitter Agents
MeSH PA D011619 Psychotropic Drugs
MeSH PA D014149 Tranquilizing Agents

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

SpeciesUseRelation
Cats For restraint or for anesthesia combined with muscle relaxation Indication
Dogs Anesthesia Indication

🐶 Veterinary products

ProductApplicantIngredients
Telazol Zoetis Inc. 2
Tzed Dechra Veterinary Products LLC 2
Zoletil for Injection Virbac AH Inc. 2

Acid dissociation constants calculated using MoKa v3.0.0

None

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

IDSource
CHEMBL2111144 ChEMBL_ID
DB11555 DRUGBANK_ID
018535 NDDF
018536 NDDF
D015041 MESH_DESCRIPTOR_UI
C0043513 UMLSCUI
CHEMBL2107559 ChEMBL_ID
3311 INN_ID
782179001 SNOMEDCT_US
96227004 SNOMEDCT_US
33754-49-3 SECONDARY_CAS_RN
D06377 KEGG_DRUG
35775 PUBCHEM_CID
1535252 RXNORM
G1R474U58U UNII

Pharmaceutical products:

None