DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
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Download
L1000
FAQ
Scroll
Substructure SMILES Example:
n1cnccc1
oclacitinib 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
Janus kinase inhibitors, antineoplastics
5589
1208319-26-9
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
oclacitinib
Molecular weight: 337.44
Formula: C15H23N5O2S
CLOGP: 1.77
LIPINSKI: 0
HAC: 7
HDO: 2
TPSA: 90.98
ALOGS: -3.26
ROTB: 4
Drug dosage:
None
ADMET properties:
None
Approvals:
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Date
Agency
Company
Orphan
None
FDA
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
None
Drug Use
| Suggest Off label Use Form|
|View source of the data|
None
🐶 Veterinary Drug Use
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Species
Use
Relation
Dogs
Pruritus associated with allergic dermatitis
Indication
Dogs
Atopic dermatitis
Indication
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🐶 Veterinary products
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Product
Applicant
Ingredients
apoquel
Zoetis Inc.
1
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Acid dissociation constants calculated using MoKa v3.0.0
None
Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Tyrosine-protein kinase JAK3
Kinase
P52333
JAK3_HUMAN
INHIBITOR
IC50
7.02
IUPHAR
Tyrosine-protein kinase JAK1
Kinase
P23458
JAK1_HUMAN
INHIBITOR
IC50
8.02
IUPHAR
Tyrosine-protein kinase JAK2
Kinase
O60674
JAK2_HUMAN
INHIBITOR
IC50
7.76
IUPHAR
Non-receptor tyrosine-protein kinase TYK2
Kinase
P29597
TYK2_HUMAN
INHIBITOR
IC50
7.12
IUPHAR
Tyrosine-protein kinase JAK2
Kinase
O60674
JAK2_HUMAN
INHIBITOR
IC50
7.76
IUPHAR
Non-receptor tyrosine-protein kinase TYK2
Kinase
P29597
TYK2_HUMAN
INHIBITOR
IC50
7.12
IUPHAR
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External reference:
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ID
Source
017725
NDDF
1487006
RXNORM
44631938
PUBCHEM_CID
9469
INN_ID
9696
IUPHAR_LIGAND_ID
99GS5XTB51
UNII
C3700984
UMLSCUI
C588062
MESH_SUPPLEMENTAL_RECORD_UI
CHEMBL2103874
ChEMBL_ID
D10141
KEGG_DRUG
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Pharmaceutical products:
None
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oclacitinib