DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
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L1000
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All
FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
saroglitazar 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
dual peroxisome proliferator activated receptors-alpha and gamma(PPAR-alpha,gamma) agonists
5047
495399-09-2
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
saroglitazar
lipaglyn
ZYH1
saroglitazar magnesium
a PPARalpha and PPARgamma agonist
Molecular weight: 439.57
Formula: C25H29NO4S
CLOGP: 5.87
LIPINSKI: 1
HAC: 5
HDO: 1
TPSA: 60.69
ALOGS: -5.47
ROTB: 11
Drug dosage:
None
ADMET properties:
None
Approvals:
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Date
Agency
Company
Orphan
June 26, 2013
CDSCO (INDIA)
CADILA HEALTHCARE
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
CHEBI has role
CHEBI:35526
antidiabetic
CHEBI has role
CHEBI:70782
PPAR-alpha agonist
CHEBI has role
CHEBI:71554
PPARgamma agonist
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Diabetic dyslipidemia associated with type 2 diabetes mellitus
indication
761000119102
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
3.58
acidic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Peroxisome proliferator-activated receptor alpha
Nuclear hormone receptor
Q07869
PPARA_HUMAN
AGONIST
EC50
9.19
SCIENTIFIC LITERATURE
SCIENTIFIC LITERATURE
Peroxisome proliferator-activated receptor gamma
Nuclear hormone receptor
P37231
PPARG_HUMAN
AGONIST
EC50
8.52
SCIENTIFIC LITERATURE
SCIENTIFIC LITERATURE
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External reference:
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entries
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ID
Source
1163258006
SNOMEDCT_US
1172675002
SNOMEDCT_US
1639792-20-3
SECONDARY_CAS_RN
60151560
PUBCHEM_CID
9677
INN_ID
C000588741
MESH_SUPPLEMENTAL_RECORD_UI
C3852920
UMLSCUI
CHEBI:134708
CHEBI
CHEMBL4297530
ChEMBL_ID
DB13115
DRUGBANK_ID
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Pharmaceutical products:
None
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saroglitazar