DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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Structure 🔎
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
Scroll
Substructure SMILES Example:
n1cnccc1
anagliptin 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
dipeptidyl aminopeptidase-IV inhibitors
4896
739366-20-2
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
anagliptin HCl
anagliptin
beskoa
anagliptin hydrochloride
suiny
anagliptin hydrochloride salt is the active compound
Molecular weight: 383.46
Formula: C19H25N7O2
CLOGP: 1.17
LIPINSKI: 0
HAC: 9
HDO: 2
TPSA: 115.42
ALOGS: -3.33
ROTB: 6
Drug dosage:
None
ADMET properties:
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Property
Value
Reference
fu (Fraction unbound in plasma)
0.77 %
Kawashima H, Watanabe R, Esaki T, Kuroda M, Nagao C, Natsume-Kitatani Y, Ohashi R, Komura H, Mizuguchi K
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Approvals:
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Date
Agency
Company
Orphan
Sept. 28, 2012
PMDA
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
MeSH PA
D054873
Dipeptidyl-Peptidase IV Inhibitors
MeSH PA
D004791
Enzyme Inhibitors
MeSH PA
D007004
Hypoglycemic Agents
MeSH PA
D011480
Protease Inhibitors
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Diabetes mellitus type 2
indication
44054006
DOID:9352
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
12.32
acidic
pKa2
5.05
Basic
pKa3
4.34
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Dipeptidyl peptidase 4
Enzyme
P27487
DPP4_HUMAN
INHIBITOR
IC50
8.42
SCIENTIFIC LITERATURE
SCIENTIFIC LITERATURE
Prolyl endopeptidase FAP
Enzyme
Q12884
SEPR_HUMAN
IC50
4.14
CHEMBL
Dipeptidyl peptidase 8
Enzyme
Q6V1X1
DPP8_HUMAN
IC50
7.17
SCIENTIFIC LITERATURE
Dipeptidyl peptidase 9
Enzyme
Q86TI2
DPP9_HUMAN
IC50
7.22
SCIENTIFIC LITERATURE
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External reference:
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ID
Source
SKK
PDB_CHEM_ID
11582
IUPHAR_LIGAND_ID
44513473
PUBCHEM_CID
9246
INN_ID
C3272640
UMLSCUI
C583175
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:136043
CHEBI
CHEMBL1929387
ChEMBL_ID
CHEMBL1929396
ChEMBL_ID
D09780
KEGG_DRUG
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Pharmaceutical products:
None
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anagliptin