palmidrol 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |
| Stem definition | Drug id | CAS RN |
|---|---|---|
| 2045 | 544-31-0 |
Description:
| Molecule | Description |
|---|---|
|
Synonyms:
|
a cannabinoid receptor-inactive eCB-related molecule used as prophylactic in helping to prevent respiratory viral infection; structure
|
Drug dosage:
None
ADMET properties:
None
Approvals:
None
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
| Source | Code | Description |
|---|---|---|
| MeSH PA | D000700 | Analgesics |
| MeSH PA | D018712 | Analgesics, Non-Narcotic |
| MeSH PA | D000890 | Anti-Infective Agents |
| MeSH PA | D000893 | Anti-Inflammatory Agents |
| MeSH PA | D000894 | Anti-Inflammatory Agents, Non-Steroidal |
| MeSH PA | D018501 | Antirheumatic Agents |
| MeSH PA | D000998 | Antiviral Agents |
| MeSH PA | D063386 | Cannabinoid Receptor Agonists |
| MeSH PA | D063385 | Cannabinoid Receptor Modulators |
| MeSH PA | D002491 | Central Nervous System Agents |
| MeSH PA | D006728 | Hormones |
| MeSH PA | D018377 | Neurotransmitter Agents |
| MeSH PA | D018373 | Peripheral Nervous System Agents |
| MeSH PA | D018689 | Sensory System Agents |
| CHEBI has role | CHEBI:35472 | anti-inflammatory drugs |
| CHEBI has role | CHEBI:35623 | anticonvulsants |
| CHEBI has role | CHEBI:35674 | antihypertensive drugs |
| CHEBI has role | CHEBI:63726 | neuroprotective agents |
Drug Use | Suggest Off label Use Form| |View source of the data|
None
🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
| Dissociation level | Dissociation constant | Type (acidic/basic) |
|---|---|---|
| pKa1 | 12.71 | acidic |
Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
| Target | Class | Pharos | UniProt | Action | Type | Activity value (-log[M]) | Mechanism action | Bioact source | MoA source |
|---|---|---|---|---|---|---|---|---|---|
| Cannabinoid receptor 1 | GPCR | Ki | 5.30 | PDSP | |||||
| Cannabinoid receptor 2 | GPCR | Ki | 5.30 | PDSP | |||||
| G-protein coupled receptor 55 | GPCR | AGONIST | EC50 | 8.40 | IUPHAR | ||||
| Fatty-acid amide hydrolase 1 | Enzyme | IC50 | 5.30 | CHEMBL |
External reference:
| ID | Source |
|---|---|
| D08328 | KEGG_DRUG |
| C0069964 | UMLSCUI |
| CHEBI:71464 | CHEBI |
| CHEMBL417675 | ChEMBL_ID |
| DB14043 | DRUGBANK_ID |
| C005958 | MESH_SUPPLEMENTAL_RECORD_UI |
| 4671 | PUBCHEM_CID |
| 871 | INN_ID |
| 6R8T1UDM3V | UNII |
| 2001986 | RXNORM |
| 011010 | NDDF |
Pharmaceutical products:
None