DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
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L1000
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All
FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
oxitropium 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
atropine derivatives
2022
99571-64-9
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
oxitropium iodide
oxytropium bromide
oxitropium
oxitropium bromide
Molecular weight: 332.42
Formula: C19H26NO4
CLOGP: -2.15
LIPINSKI: 0
HAC: 5
HDO: 1
TPSA: 59.06
ALOGS: -4.76
ROTB: 6
Drug dosage:
Dose
Unit
Route
0.60
mg
Inhal.aerosol
4
mg
Inhal.solution
ADMET properties:
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Property
Value
Reference
BA (Bioavailability)
1 %
Kim MT, Sedykh A, Chakravarti SK, Saiakhov RD, Zhu H
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Approvals:
None
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
R03BB02
RESPIRATORY SYSTEM
DRUGS FOR OBSTRUCTIVE AIRWAY DISEASES
OTHER DRUGS FOR OBSTRUCTIVE AIRWAY DISEASES, INHALANTS
Anticholinergics
MeSH PA
D010276
Parasympatholytics
MeSH PA
D018373
Peripheral Nervous System Agents
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Chronic obstructive lung disease
indication
13645005
DOID:3083
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
13.24
acidic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
None
External reference:
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ID
Source
004014
NDDF
006120
NDDF
30286-75-0
SECONDARY_CAS_RN
32649
RXNORM
349953003
SNOMEDCT_US
3955
INN_ID
395816001
SNOMEDCT_US
395993006
SNOMEDCT_US
6917866
PUBCHEM_CID
8G15T83E6I
UNII
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Pharmaceutical products:
None
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oxitropium