dimethisterone 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
steroids, progestogens 904 79-64-1

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • dimethisterone
  • dimethiderome
  • dimethisteron
A synthetic progestational hormone without significant estrogenic or androgenic properties. It was formerly used as the progestational component in SEQUENTIAL ORAL CONTRACEPTIVE AGENTS .
  • Molecular weight: 340.51
  • Formula: C23H32O2
  • CLOGP: 4.16
  • LIPINSKI: 0
  • HAC: 2
  • HDO: 1
  • TPSA: 37.30
  • ALOGS: -5.28
  • ROTB: 1

Drug dosage:

None

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

SourceCodeDescription
CHEBI has role CHEBI:50113 androgene
MeSH PA D003270 Contraceptive Agents
MeSH PA D003271 Contraceptive Agents, Female
MeSH PA D000080066 Contraceptive Agents, Hormonal
MeSH PA D003278 Contraceptives, Oral, Hormonal
MeSH PA D003280 Contraceptives, Oral, Synthetic
MeSH PA D012102 Reproductive Control Agents

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

None

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

IDSource
D02298 KEGG_DRUG
C0012391 UMLSCUI
CHEBI:4606 CHEBI
CHEMBL3989718 ChEMBL_ID
CHEMBL2106347 ChEMBL_ID
D004116 MESH_DESCRIPTOR_UI
6607 PUBCHEM_CID
K4MZ02M175 UNII
001301 NDDF
41354-30-7 SECONDARY_CAS_RN

Pharmaceutical products:

None