DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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Structure 🔎
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
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All
FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
cytisine 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
5217
485-35-8
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
cytisine
baptitoxine
tabex
RN given refers to (R)-isomer; structure
Molecular weight: 190.25
Formula: C11H14N2O
CLOGP: -0.41
LIPINSKI: 0
HAC: 3
HDO: 1
TPSA: 32.34
ALOGS: -1.37
ROTB: 0
Drug dosage:
None
ADMET properties:
None
Approvals:
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Date
Agency
Company
Orphan
None
Health Canada
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
CHEBI has role
CHEBI:38231
phytotoxins
CHEBI has role
CHEBI:47958
muscarinic agonists
CHEBI has role
CHEBI:76924
plant metabolites
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Smoking cessation assistance
indication
384742004
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
8.18
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Neuronal acetylcholine receptor subunit alpha-7
Ion channel
P36544
ACHA7_HUMAN
Ki
5.85
CHEMBL
Acetylcholine receptor subunit delta
Ion channel
ACHD_TORCA
EC50
4
CHEMBL
Neuronal acetylcholine receptor subunit alpha-4
Ion channel
ACHA4_RAT
Ki
9.47
CHEMBL
Neuronal acetylcholine receptor subunit alpha-7
Ion channel
ACHA7_RAT
Ki
9.05
CHEMBL
Acetylcholine receptor subunit alpha
Ion channel
ACHA_TORCA
IC50
5.45
CHEMBL
Nicotinic acetylcholine receptor alpha 5 subunit
Ion channel
A9XFY4_MUSDO
Ki
5.91
CHEMBL
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External reference:
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entries
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ID
Source
C5E
PDB_CHEM_ID
10235
PUBCHEM_CID
11015
INN_ID
1723152
RXNORM
1ZI8CA9FWW
UNII
5347
IUPHAR_LIGAND_ID
53S5U404NU
UNII
76283008
SNOMEDCT_US
C004712
MESH_SUPPLEMENTAL_RECORD_UI
C0056913
UMLSCUI
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Pharmaceutical products:
None
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cytisine