clobenztropine 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
atropine derivatives 3715 5627-46-3

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • clobenztropine
  • teprin
  • Molecular weight: 341.88
  • Formula: C21H24ClNO
  • CLOGP: 4.23
  • LIPINSKI: 0
  • HAC: 2
  • HDO: 0
  • TPSA: 12.47
  • ALOGS: -5.77
  • ROTB: 4

Drug dosage:

None

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

None

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 9.86 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

TargetClassPharosUniProtActionTypeActivity value
(-log[M])		Mechanism
action		Bioact sourceMoA source
Sodium-dependent dopamine transporter Transporter Ki 7.52 CHEMBL

External reference:

IDSource
C5420916 UMLSCUI
CHEBI:135452 CHEBI
CHEMBL2146132 ChEMBL_ID
1687 PUBCHEM_CID
1388 INN_ID
M8CDT278F8 UNII

Pharmaceutical products:

None