mestanolone 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
androgens/anabolic steroids 3341 521-11-9

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • mestaline
  • mesanolon
  • mestanolone
  • mestalone
  • mestanolon
  • methylandrostanolone
  • methylantalon
non-virilizing androgenic steroid; RN given refers to (5alpha,17beta)-isomer; structure
  • Molecular weight: 304.47
  • Formula: C20H32O2
  • CLOGP: 4.07
  • LIPINSKI: 0
  • HAC: 2
  • HDO: 1
  • TPSA: 37.30
  • ALOGS: -4.90
  • ROTB: 0

Drug dosage:

None

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

None

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

None

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

TargetClassPharosUniProtActionTypeActivity value
(-log[M])
Mechanism
action
Bioact sourceMoA source
Androgen receptor Nuclear hormone receptor AGONIST KEGG DRUG KEGG DRUG
Sex hormone-binding globulin Secreted Kd 8.81 CHEMBL

External reference:

IDSource
D01533 KEGG_DRUG
C0066031 UMLSCUI
CHEBI:31825 CHEBI
CHEMBL261514 ChEMBL_ID
C008376 MESH_SUPPLEMENTAL_RECORD_UI
10633 PUBCHEM_CID
862 INN_ID
S712YZ168E UNII

Pharmaceutical products:

None