sulforidazine 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
2532 14759-06-9

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • sulforidazine
  • imagotan
  • inofal
  • psychoson
  • sulphoridazine
  • thioridazine-2-sulfone
  • Molecular weight: 402.57
  • Formula: C21H26N2O2S2
  • CLOGP: 4.62
  • LIPINSKI: 0
  • HAC: 4
  • HDO: 0
  • TPSA: 40.62
  • ALOGS: -4.65
  • ROTB: 4

Drug dosage:

None

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

SourceCodeDescription
MeSH PA D000928 Antidepressive Agents
MeSH PA D014150 Antipsychotic Agents
MeSH PA D002491 Central Nervous System Agents
MeSH PA D002492 Central Nervous System Depressants
MeSH PA D011619 Psychotropic Drugs
MeSH PA D014149 Tranquilizing Agents

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 9.22 Basic
pKa2 3.45 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

TargetClassPharosUniProtActionTypeActivity value
(-log[M])
Mechanism
action
Bioact sourceMoA source
D(2) dopamine receptor GPCR Ki 9.61 PDSP
D(3) dopamine receptor GPCR Ki 9.16 PDSP

External reference:

IDSource
C0075591 UMLSCUI
CHEBI:135644 CHEBI
CHEMBL2107268 ChEMBL_ID
C040634 MESH_SUPPLEMENTAL_RECORD_UI
C476405 MESH_SUPPLEMENTAL_RECORD_UI
31765 PUBCHEM_CID
2394 INN_ID
B7599I244X UNII
725620001 SNOMEDCT_US

Pharmaceutical products:

None