DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
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Smart API
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L1000
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FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
anhydrovinblastine 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
vinca alkaloids
219
38390-45-3
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
anhydrovinblastine
anhydrovincaleukoblastine
Molecular weight: 792.97
Formula: C46H56N4O8
CLOGP: 5.19
LIPINSKI: 3
HAC: 12
HDO: 2
TPSA: 133.87
ALOGS: -5.01
ROTB: 10
Drug dosage:
None
ADMET properties:
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Property
Value
Reference
t_half (Half-life)
18 hours
Lombardo F, Berellini G, Obach RS
CL (Clearance)
12 mL/min/kg
Lombardo F, Berellini G, Obach RS
Vd (Volume of distribution)
12 L/kg
Lombardo F, Berellini G, Obach RS
S (Water solubility)
10 mg/mL
Benet LZ, Broccatelli F, Oprea TI
BDDCS (Biopharmaceutical Drug Disposition Classification System)
1
Benet LZ, Broccatelli F, Oprea TI
EoM (Fraction excreted unchanged in urine)
0.50 %
Benet LZ, Broccatelli F, Oprea TI
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Approvals:
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Date
Agency
Company
Orphan
Jan. 1, 1965
YEAR INTRODUCED
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
None
Drug Use
| Suggest Off label Use Form|
|View source of the data|
None
🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
11.32
acidic
pKa2
13.81
acidic
pKa3
7.58
Basic
pKa4
6.94
Basic
pKa5
6.11
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Multidrug resistance protein 1
Transporter
P08183
MDR1_HUMAN
WOMBAT-PK
Canalicular multispecific organic anion transporter 1
Transporter
Q92887
MRP2_HUMAN
WOMBAT-PK
Multidrug resistance-associated protein 1
Transporter
P33527
MRP1_HUMAN
WOMBAT-PK
Multidrug resistance-associated protein 7
Transporter
Q5T3U5
MRP7_HUMAN
WOMBAT-PK
Tubulin beta-4B chain
Structural
P68371
TBB4B_HUMAN
WOMBAT-PK
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External reference:
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ID
Source
11104750
PUBCHEM_CID
5B622U08B3
UNII
C0796616
UMLSCUI
CHEBI:1322
CHEBI
DB12586
DRUGBANK_ID
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Pharmaceutical products:
None
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anhydrovinblastine