moxastine 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
antihistaminics 1852 3572-74-5

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • alfadryl
  • moxastine
  • mephenhydramine
  • moxastin
  • theoclan moxastin
  • mephenhydramine theoclate
  • mephenhydrinate
  • moxastine theoclate
  • Molecular weight: 269.39
  • Formula: C18H23NO
  • CLOGP: 3.85
  • LIPINSKI: 0
  • HAC: 2
  • HDO: 0
  • TPSA: 12.47
  • ALOGS: -3.92
  • ROTB: 6

Drug dosage:

None

ADMET properties:

None

Approvals:

None

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

None

Drug Use | Suggest Off label Use Form| |View source of the data|

None




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 8.56 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

TargetClassPharosUniProtActionTypeActivity value
(-log[M])		Mechanism
action		Bioact sourceMoA source
Histamine H1 receptor GPCR ANTAGONIST SCIENTIFIC LITERATURE SCIENTIFIC LITERATURE

External reference:

IDSource
C1881908 UMLSCUI
CHEBI:135108 CHEBI
CHEMBL1742465 ChEMBL_ID
19142 PUBCHEM_CID
C008553 MESH_SUPPLEMENTAL_RECORD_UI
1791 INN_ID
ZSJ254W6SF UNII

Pharmaceutical products:

None