falecalcitriol 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |

Stem definitionDrug idCAS RN
Vitamin D analogues/derivatives 1127 83805-11-2

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • ST-630
  • fulstan
  • hornel
  • falecalcitriol
  • flocacitriol
  • flocalcitriol
  • flocalcitrol
  • falecalcitoriol
  • Molecular weight: 524.59
  • Formula: C27H38F6O3
  • CLOGP: 6.96
  • LIPINSKI: 2
  • HAC: 3
  • HDO: 3
  • TPSA: 60.69
  • ALOGS: -5.43
  • ROTB: 8

Drug dosage:

None

ADMET properties:

None

Approvals:

DateAgencyCompanyOrphan
April 4, 2001 PMDA Taisho Pharmaceutical

FDA Adverse Event Reporting System (Female)

None

FDA Adverse Event Reporting System (Male)

None

FDA Adverse Event Reporting System (Geriatric)

None

FDA Adverse Event Reporting System (Pediatric)

None

Pharmacologic Action:

SourceCodeDescription
MeSH PA D003879 Dermatologic Agents

Drug Use | Suggest Off label Use Form| |View source of the data|

DiseaseRelationSNOMED_IDDOID
Osteomalacia indication 4598005 DOID:10573
Hypoparathyroidism indication 36976004 DOID:11199
Rickets indication 41345002 DOID:10609




🐶 Veterinary Drug Use

None

🐶 Veterinary products

None

Acid dissociation constants calculated using MoKa v3.0.0

Dissociation levelDissociation constantType (acidic/basic)
pKa1 10.91 acidic
pKa2 13.7 acidic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

IDSource
D01662 KEGG_DRUG
C0046706 UMLSCUI
CHEBI:31590 CHEBI
CHEMBL2106158 ChEMBL_ID
C040488 MESH_SUPPLEMENTAL_RECORD_UI
2781 IUPHAR_LIGAND_ID
7103 INN_ID
G70A8514T8 UNII
5282190 PUBCHEM_CID

Pharmaceutical products:

None