azanidazole indications/contra

Stem definitionDrug idCAS RN
antiprotozoals and radiosensitizers, metronidazole derivatives 264 62973-76-6

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • azanidazole
  • nitromidine
  • Molecular weight: 246.23
  • Formula: C10H10N6O2
  • CLOGP: 0.33
  • LIPINSKI: 0
  • HAC: 8
  • HDO: 1
  • TPSA: 115.44
  • ALOGS: -2.49
  • ROTB: 3

Drug dosage:

None

Approvals:

None

FDA Adverse Event Reporting System

None

Pharmacologic Action:

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SourceCodeDescription
ATC G01AF13 GENITO URINARY SYSTEM AND SEX HORMONES
GYNECOLOGICAL ANTIINFECTIVES AND ANTISEPTICS
ANTIINFECTIVES AND ANTISEPTICS, EXCL. COMBINATIONS WITH CORTICOSTEROIDS
Imidazole derivatives
ATC P01AB04 ANTIPARASITIC PRODUCTS, INSECTICIDES AND REPELLENTS
ANTIPROTOZOALS
AGENTS AGAINST AMOEBIASIS AND OTHER PROTOZOAL DISEASES
Nitroimidazole derivatives

Drug Use (View source of the data)

None

Acid dissociation constants calculated using MoKa v3.0.0

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Dissociation levelDissociation constantType (acidic/basic)
pKa1 4.56 Basic
pKa2 2.1 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

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IDSource
D03028 KEGG_DRUG
6436171 PUBCHEM_CID
CHEMBL134920 ChEMBL_ID
CHEBI:135001 CHEBI
C023624 MESH_SUPPLEMENTAL_RECORD_UI
YP2Y0DRX4S UNII
4274 INN_ID

Pharmaceutical products:

None