Beta-2 adrenergic receptor

Description:

Description
  • Accession: Q28044
  • Swissprot: ADRB2_BOVIN
  • Organism: Bos taurus
  • Gene: ADRB2
  • Target class: GPCR

Drug Relations:

alprenolol
One of the ADRENERGIC BETA-ANTAGONISTS used as an antihypertensive, anti-anginal, and anti-arrhythmic agent. Bioactivity details MOA
betaxolol
A cardioselective beta-1-adrenergic antagonist with no partial agonist activity. Bioactivity details MOA
clenbuterol
A substituted phenylaminoethanol that has beta-2 adrenomimetic properties at very low doses. It is used as a bronchodilator in asthma. Bioactivity details MOA
isoprenaline
Isopropyl analog of EPINEPHRINE; beta-sympathomimetic that acts on the heart, bronchi, skeletal muscle, alimentary tract, etc. It is used mainly as bronchodilator and heart stimulant. Bioactivity details MOA
nifenalol
adrenergic beta-blocker with good antiarrhythmic properties; also tends to lower blood pressure & provide protection against angina; minor descriptor (75-86); on-line & INDEX MEDICUS search ETHANOLAMINES (75-86); RN given refers to parent cpd without isomeric designation Bioactivity details MOA
norepinephrine
Precursor of epinephrine that is secreted by the ADRENAL MEDULLA and is a widespread central and autonomic neurotransmitter. Norepinephrine is the principal transmitter of most postganglionic sympathetic fibers, and of the diffuse projection system in the brain that arises from the LOCUS CERULEUS. It is also found in plants and is used pharmacologically as a sympathomimetic. Bioactivity details MOA
orciprenaline
A beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM. Bioactivity details MOA
practolol
A beta-1 adrenergic antagonist that has been used in the emergency treatment of CARDIAC ARRYTHMIAS. Bioactivity details MOA
prenalterol
A partial adrenergic agonist with functional beta 1-receptor specificity and inotropic effect. It is effective in the treatment of acute CARDIAC FAILURE, postmyocardial infarction low-output syndrome, SHOCK, and reducing ORTHOSTATIC HYPOTENSION in the SHY-RAGER SYNDROME. Bioactivity details MOA
pronetalol
Bioactivity details MOA
propranolol
A widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse effects instigate replacement by newer drugs. Bioactivity details MOA
salbutamol
A short-acting beta-2 adrenergic agonist that is primarily used as a bronchodilator agent to treat ASTHMA. Albuterol is prepared as a racemic mixture of R(-) and S(+) stereoisomers. The stereospecific preparation of R(-) isomer of albuterol is referred to as levalbuterol. Bioactivity details MOA
sotalol
An adrenergic beta-antagonist that is used in the treatment of life-threatening arrhythmias. Bioactivity details MOA
terbutaline
A selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic. Bioactivity details MOA
toliprolol
was MH 1975-92 (see under PROPANOLAMINES 1981-90, was DOBEROL see under PROPANOLAMINES 1975-80); KOE 592 was see TOLIPROLOL 1975-92; use PROPANOLAMINES to search TOLIPROLOL 1975-92; beta adrenergic blockader with some stimulant action; it has been proposed for angina pectoris Bioactivity details MOA
tulobuterol
Bioactivity details MOA