acetarsol indications/contra

Stem definitionDrug idCAS RN
55 97-44-9

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • acetarsol
  • acetarsone
  • acetphenarsine
  • arsaphen
  • Molecular weight: 275.09
  • Formula: C8H10AsNO5
  • CLOGP: -1.36
  • LIPINSKI: 0
  • HAC: 6
  • HDO: 4
  • TPSA: 106.86
  • ALOGS: -1.99
  • ROTB: 2

Drug dosage:

DoseUnitRoute
0.50 g V

Approvals:

None

FDA Adverse Event Reporting System

None

Pharmacologic Action:

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SourceCodeDescription
ATC A07AX02 ALIMENTARY TRACT AND METABOLISM
ANTIDIARRHEALS, INTESTINAL ANTIINFLAMMATORY/ANTIINFECTIVE AGENTS
INTESTINAL ANTIINFECTIVES
Other intestinal antiinfectives
ATC G01AB01 GENITO URINARY SYSTEM AND SEX HORMONES
GYNECOLOGICAL ANTIINFECTIVES AND ANTISEPTICS
ANTIINFECTIVES AND ANTISEPTICS, EXCL. COMBINATIONS WITH CORTICOSTEROIDS
Arsenic compounds
ATC P01CD02 ANTIPARASITIC PRODUCTS, INSECTICIDES AND REPELLENTS
ANTIPROTOZOALS
AGENTS AGAINST LEISHMANIASIS AND TRYPANOSOMIASIS
Arsenic compounds
MeSH PA D000890 Anti-Infective Agents

Drug Use (View source of the data)

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DiseaseRelationSNOMED_IDDOID
Amebic infection indication 111910009 DOID:9181

Acid dissociation constants calculated using MoKa v3.0.0

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Dissociation levelDissociation constantType (acidic/basic)
pKa1 3.84 acidic
pKa2 8.4 acidic
pKa3 9.83 acidic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

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IDSource
D07110 KEGG_DRUG
806529YU1N UNII
371 INN_ID
1985 PUBCHEM_CID
421639009 SNOMEDCT_US
22236007 SNOMEDCT_US
005948 NDDF
CHEBI:135135 CHEBI
CHEMBL1330792 ChEMBL_ID
C005284 MESH_SUPPLEMENTAL_RECORD_UI

Pharmaceutical products:

None