caroverine indications/contra

Stem definitionDrug idCAS RN
spasmolytics with a papaverine-like action 514 23465-76-1

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • caroverine
  • spadon
  • Molecular weight: 365.48
  • Formula: C22H27N3O2
  • CLOGP: 4.11
  • LIPINSKI: 0
  • HAC: 5
  • HDO: 0
  • TPSA: 45.14
  • ALOGS: -4.09
  • ROTB: 8

Drug dosage:

None

Approvals:

None

FDA Adverse Event Reporting System

None

Pharmacologic Action:

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SourceCodeDescription
ATC A03AX11 ALIMENTARY TRACT AND METABOLISM
DRUGS FOR FUNCTIONAL GASTROINTESTINAL DISORDERS
DRUGS FOR FUNCTIONAL GASTROINTESTINAL DISORDERS
Other drugs for functional gastrointestinal disorders
MeSH PA D002121 Calcium Channel Blockers
MeSH PA D002317 Cardiovascular Agents
MeSH PA D018683 Excitatory Amino Acid Agents
MeSH PA D018691 Excitatory Amino Acid Antagonists
MeSH PA D049990 Membrane Transport Modulators
MeSH PA D018377 Neurotransmitter Agents

Drug Use (View source of the data)

None

Acid dissociation constants calculated using MoKa v3.0.0

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Dissociation levelDissociation constantType (acidic/basic)
pKa1 9.16 Basic
pKa2 1.8 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

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IDSource
D07098 KEGG_DRUG
65709 PUBCHEM_CID
CHEMBL1729803 ChEMBL_ID
XJ73B0K6KB UNII
3254 INN_ID
C000957 MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:135541 CHEBI

Pharmaceutical products:

None