DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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Structure 🔎
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
Redial
About
Download
L1000
FAQ
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All
FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
lobeglitazone 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
peroxisome proliferator activating receptor-gamma (PPAR-gamma) agonists, thiazolidinedione derivatives
5078
607723-33-1
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
lobeglitazone
lobeglitazone sulfate
CKD-501
duvie
putative antidiabetic agent for type 2 diabetes
Molecular weight: 480.54
Formula: C24H24N4O5S
CLOGP: 4.37
LIPINSKI: 0
HAC: 9
HDO: 1
TPSA: 102.88
ALOGS: -4.42
ROTB: 10
Drug dosage:
Dose
Unit
Route
0.50
mg
O
ADMET properties:
None
Approvals:
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Date
Agency
Company
Orphan
July 4, 2013
Korean Food and Drug Administration (KFDA)
Chong Kun Dang
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1
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FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
A10BD26
ALIMENTARY TRACT AND METABOLISM
DRUGS USED IN DIABETES
BLOOD GLUCOSE LOWERING DRUGS, EXCL. INSULINS
Combinations of oral blood glucose lowering drugs
ATC
A10BG04
ALIMENTARY TRACT AND METABOLISM
DRUGS USED IN DIABETES
BLOOD GLUCOSE LOWERING DRUGS, EXCL. INSULINS
Thiazolidinediones
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
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Disease
Relation
SNOMED_ID
DOID
Diabetes mellitus type 2
indication
44054006
DOID:9352
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🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
6.33
acidic
pKa2
5.62
Basic
pKa3
1.02
Basic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Peroxisome proliferator-activated receptor gamma
Nuclear hormone receptor
P37231
PPARG_HUMAN
AGONIST
EC50
7.75
SCIENTIFIC LITERATURE
SCIENTIFIC LITERATURE
Peroxisome proliferator-activated receptor alpha
Nuclear hormone receptor
Q07869
PPARA_HUMAN
AGONIST
EC50
7.70
SCIENTIFIC LITERATURE
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External reference:
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ID
Source
8LX
PDB_CHEM_ID
763108-62-9
SECONDARY_CAS_RN
8729
INN_ID
9826451
PUBCHEM_CID
C2744790
UMLSCUI
C546215
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:136052
CHEBI
CHEMBL3585580
ChEMBL_ID
CHEMBL3780740
ChEMBL_ID
DB09198
DRUGBANK_ID
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Pharmaceutical products:
None
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Structure 🔎
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L1000
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lobeglitazone