DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
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Structure 🔎
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L1000
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DrugCentral 2023 🐕
2022 Update-Veterinary Drugs & Uses
Search
Structure 🔎
Similarity 🔎
Smart API
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L1000
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FDA-approved
EMA-approved
PMDA-approved
Target Card Uniprot Example:
P23975
ridaforolimus 🐶
Veterinary Use |
Indications/Contra
| FAERs-F
| FAERs-M
| Orange Bk
| BioActivity |
Stem definition
Drug id
CAS RN
immunosuppressants, rapamycin derivatives
4778
572924-54-0
Description:
Molecule
Description
Molfile
Inchi
Smiles
Synonyms:
deforolimus
ridaforolimus
AP23573
MK-8669
jenzyl
an mTOR inhibitor for the treatment of cancer
Molecular weight: 990.22
Formula: C53H84NO14P
CLOGP: 7.20
LIPINSKI: 3
HAC: 15
HDO: 2
TPSA: 201.50
ALOGS: -6.09
ROTB: 8
Drug dosage:
None
ADMET properties:
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Property
Value
Reference
t_half (Half-life)
46.30 hours
Lombardo F, Berellini G, Obach RS
Vd (Volume of distribution)
3.20 L/kg
Lombardo F, Berellini G, Obach RS
CL (Clearance)
1.10 mL/min/kg
Lombardo F, Berellini G, Obach RS
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Approvals:
None
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
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Source
Code
Description
ATC
L01EG03
ANTINEOPLASTIC AND IMMUNOMODULATING AGENTS
ANTINEOPLASTIC AGENTS
PROTEIN KINASE INHIBITORS
Mammalian target of rapamycin (mTOR) kinase inhibitors
CHEBI has role
CHEBI:35610
antineoplastic agents
CHEBI has role
CHEBI:68481
mTOR inhibitors
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Drug Use
| Suggest Off label Use Form|
|View source of the data|
None
🐶 Veterinary Drug Use
None
🐶 Veterinary products
None
Acid dissociation constants calculated using MoKa v3.0.0
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Dissociation level
Dissociation constant
Type (acidic/basic)
pKa1
10.5
acidic
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Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
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Target
Class
Pharos
UniProt
Action
Type
Activity value
(-log[M])
Mechanism
action
Bioact source
MoA source
Serine/threonine-protein kinase mTOR
Kinase
P42345
MTOR_HUMAN
INHIBITOR
IC50
9.70
SCIENTIFIC LITERATURE
SCIENTIFIC LITERATURE
Dual specificity tyrosine-phosphorylation-regulated kinase 1B
Kinase
Q9Y463
DYR1B_HUMAN
Kd
5.90
CHEMBL
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External reference:
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ID
Source
11520894
PUBCHEM_CID
48Z35KB15K
UNII
7884
IUPHAR_LIGAND_ID
8822
INN_ID
C2713007
UMLSCUI
C515074
MESH_SUPPLEMENTAL_RECORD_UI
CHEBI:82677
CHEBI
CHEMBL2103839
ChEMBL_ID
D08900
KEGG_DRUG
DB06233
DRUGBANK_ID
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Pharmaceutical products:
None
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ridaforolimus