amezinium metilsulfate indications/contra

Stem definitionDrug idCAS RN
153 30578-37-1

Description:

MoleculeDescription

Molfile Inchi Smiles

Synonyms:

  • amezinium methyl sulfate
  • amezinium
  • amezinium metilsulfate
  • regulton
  • Molecular weight: 202.24
  • Formula: C11H12N3O
  • CLOGP: -1.48
  • LIPINSKI: 0
  • HAC: 4
  • HDO: 1
  • TPSA: 52.02
  • ALOGS: -2.38
  • ROTB: 2

Drug dosage:

DoseUnitRoute
30 mg O

Approvals:

None

FDA Adverse Event Reporting System

None

Pharmacologic Action:

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SourceCodeDescription
ATC C01CA25 CARDIOVASCULAR SYSTEM
CARDIAC THERAPY
CARDIAC STIMULANTS EXCL. CARDIAC GLYCOSIDES
Adrenergic and dopaminergic agents
MeSH PA D001337 Autonomic Agents
MeSH PA D004791 Enzyme Inhibitors
MeSH PA D008996 Monoamine Oxidase Inhibitors
MeSH PA D018373 Peripheral Nervous System Agents
MeSH PA D013566 Sympathomimetics

Drug Use (View source of the data)

None

Acid dissociation constants calculated using MoKa v3.0.0

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Dissociation levelDissociation constantType (acidic/basic)
pKa1 3.39 Basic

Orange Book patent data (new drug applications)

None

Orange Book exclusivity data (new drug applications)

None

Bioactivity Summary:

None

External reference:

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IDSource
C0051570 UMLSCUI
D01304 KEGG_DRUG
03NR868ICX UNII
4066 INN_ID
71926 PUBCHEM_CID
004308 NDDF
CHEBI:31201 CHEBI
CHEMBL2106667 ChEMBL_ID
CHEMBL2110922 ChEMBL_ID
C027784 MESH_SUPPLEMENTAL_RECORD_UI

Pharmaceutical products:

None